1354644-62-4Relevant articles and documents
Synthesis of N -azolylindoles by copper-catalyzed C-H/N-H coupling-annulation sequence of o -alkynylanilines
Oda, Yoshiro,Hirano, Koji,Satoh, Tetsuya,Miura, Masahiro
supporting information; experimental part, p. 664 - 667 (2012/02/16)
A wide range of o-alkynylanilines undergo a copper-catalyzed direct C-H/N-H coupling with azoles followed by benzannulation to form the corresponding N-azolylindoles in good yields. The domino reaction proceeds effectively with molecular oxygen as the sol