142521-09-3Relevant articles and documents
Pd-Catalyzed Indole Synthesis via C-H Activation and Bisamination Sequence with Diaziridinone
Wang, Jianjun,Sun, Xiaofeng,Hu, Daguo,Shi, Yian
supporting information, p. 7561 - 7565 (2021/10/02)
This work describes an efficient Pd-catalyzed indole synthesis. A wide variety of indoles can be obtained in good yields from readily available vinyl bromides. The reaction likely proceeds through a sequential aryl C-H activation and bisamination of a resulting pallada(II)cycle with diaziridinone.
AMIDE COMPOUND AND MEDICINAL USE THEREOF
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, (2013/02/27)
A compound of formula [I-W]: wherein each symbol is as defined in the description, or a pharmaceutically acceptable salt thereof.