1436868-42-6Relevant articles and documents
Three-component synthesis of poly-substituted tetrahydroindoles through p-TsOH promoted alkoxylation
Shi, Qing-Qing,Fu, Li-Ping,Shi, Yu,Ding, Hua-Qin,Luo, Jing-Hua,Jiang, Bo,Tu, Shu-Jiang
supporting information, p. 3176 - 3179 (2013/06/26)
Concise and efficient three-component domino reactions to highly substituted tetrahydroindole derivatives promoted by p-TsOH have been developed under microwave irradiation condition. The direct C3-alkoxylation of indole framework was achieved in a one-pot operation. The reaction proceeds at fast rates and can be finished within 30 min, which makes workup convenient to give good chemical yields.