172945-94-7Relevant articles and documents
DOUBLE-HEADED PROTEASE INHIBITOR
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Paragraph 1092; 1093; 1095, (2020/09/17)
The present invention provides a compound that is highly safe and useful in the prevention, alleviation, and/or treatment of various diseases involving enteropeptidase inhibition and/or trypsin inhibition, a pharmaceutical composition containing the compo
Nucleopeptidic bioconjugates containing a sulfamide bridge: Linkage via the Mitsunobu reaction
Criton,Dewynter,Aouf,Montero,Imbach
, p. 1795 - 1801 (2007/10/02)
The synthesis of compounds connecting unprotected 2'-deoxyribonucleosides (T,dC,dG,dA) with N-Boc sulfamoyl derivatives of natural aminoacid esters (Phe, Asp) was carried out by Mitsunobu reaction, using regiospecific coupling. The created link was a prio