176389-60-9Relevant articles and documents
Photoaffinity labeling of the ligand-interacting helix of the retinoic acid receptor alpha
Sasaki, Toru,Morisaki, Naoko,Iwasaki, Shigeo,Kagechika, Hiroshi,Fukasawa, Hiroshi,Shudo, Koichi,Shida, Yasuo,Hashimoto, Yuichi
, p. 913 - 916 (1997)
Two photoaffinity-labeling probes for retinoic acid receptor (RAR) α, 4-[(3-(3-(trifluoromethyl)-3H-diazirin-3-yl)phenyl)carboxamido]benzoic acid (3DIAM) and its para-isomer (4DIAM), were designed and synthesized. Both compounds possess high affinity for
SMALL MOLECULE MODULATORS OF PCSK9 AND METHODS OF USE THEREOF
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Paragraph 0363; 0373, (2016/02/22)
A compound of Formula (I): or a pharmaceutically acceptable salt, hydrate, solvate, or racemic mixture or stereoisomer thereof, and methods for preventing or treating an LDL-cholesterol-related disease or disorder using such compound(s), and kits and comp