186320-14-9Relevant articles and documents
Maytansinoid derivatives with peptide linker and conjugates thereof
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Page/Page column 103; 104, (2016/04/20)
The invention relates to novel cell-binding agent-cytotoxic agent conjugate having a peptide linkers and more specifically to conjugates of formula (I). The invention also provides novel cytotoxic agents of formula (II), linker compounds represented by fo
Preparation of 16β-estradiol derivative libraries as bisubstrate inhibitors of 17β-hydroxysteroid dehydrogenase type 1 using the multidetachable sulfamate linker
Berube, Marie,Delagoutte, Florian,Poirier, Donald
experimental part, p. 1590 - 1631 (2010/05/17)
Combinatorial chemistry is a powerful tool used to rapidly generate a large number of potentially biologically active compounds. In our goal to develop bisubstrate inhibitors of 17β-hydroxysteroid dehydrogenase type 1 (17β-HSD1) that interact with both th