188719-30-4Relevant articles and documents
Mustard prodrugs for activation by Escherichia coli nitroreductase in gene-directed enzyme prodrug therapy
Friedlos, Frank,Denny, William A.,Palmer, Brian D.,Springer, Caroline J.
, p. 1270 - 1275 (2007/10/03)
Twenty nitrogen mustard analogues derived from 5-(aziridin-l-yl)-2,4- dinitrobenzamide (CB 1954, 1) were evaluated as candidate prodrugs for gene- directed enzyme prodrug therapy (GDEPT) in Chinese hamster V79 cell lines engineered to express Escherichia