196195-47-8Relevant articles and documents
Non-steroidal irreversible inhibitors of aromatase based on N-pentyl-3-phenylpyrrolidine-2,5-dione
Saeed,Khodarahmi,Fradgley,Smith,Nicholls,King,Ahmadi
, p. 265 - 277 (2007/10/03)
1-Pentyl-3-(3'-propynyloxyphenyl) pyrrolidine-2,5-dione (20), its 3-propynyl substituted derivative (18), with its corresponding 4'-substituted isomer (21), constitute the first of a new type of non-steroidal mechanism-based inactivators of aromatase with