237769-03-8Relevant articles and documents
Application of oxathiazolidine-S-oxide chemistry to the large-scale single-step synthesis of an O-arylethanolamine
Barker, Alan C.,Boardman, Kay A.,Broady, Simon D.,Moss, William O.,Patel, Bharti,Senior, Michael W.,Warren, Kenneth E. H.
, p. 253 - 255 (1999)
Alternative routes to the arylethanolamine subunit of a development drug have been investigated. The selected route, involving O-alkylation of a phenol using N-benzyloxathiazolidine-S-oxide, was developed to give a process used successfully for pilot plan
Novel preparation of functionalized iodotetrahydronaphthyridine, iodoazaindoline, and iodotetrahydropyridoazepine systems
Nguyen, Hanh Nho,Wang, Zhan J.
, p. 7460 - 7463 (2008/03/14)
A novel method, which utilizes a key halogen dance step for the preparation of iodotetrahydronaphthyridine, iodoazaindoline, and iodotetrahydropyridoazepine ring-systems is described. A variety of transformations of the iodo-functional group are also repo