24469-05-4Relevant articles and documents
Easily accessible auxiliary for palladium-catalyzed intramolecular amination of C(sp2)-H and C(sp3)-H bonds at δ- And ε-Positions
Wang, Chao,Chen, Changpeng,Zhang, Jingyu,Han, Jian,Wang, Qian,Guo, Kun,Liu, Pei,Guan, Mingyu,Yao, Yingming,Zhao, Yingsheng
supporting information, p. 9884 - 9888,5 (2014/10/15)
An easily synthesized and accessible N,O-bidentate auxiliary has been developed for selective C-H activation under palladium catalysis. The novel auxiliary showed its first powerful application in C-H functionalization of remote positions. Both C(sp2)-H and C(sp3)-H bonds at δ- and ε-positions were effectively activated, thus giving tetrahydroquinolines, benzomorpholines, pyrrolidines, and indolines in moderate to excellent yields by palladium-catalyzed intramolecular C-H amination.
INHIBITORS OF UNDECAPRENYL PYROPHOSPHATE SYNTHASE
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Page/Page column 120-121, (2008/06/13)
The present invention relates to compounds that are selective and/or potent inhibitors of UPPS. In addition to compounds which inhibit UPPS, the invention also provides pharmaceutical compositions comprising these compounds and methods of using these comp
An Expedient and Practical Method for the Synthesis of A Diverse Series of Cyclopropane α-Amino Acids and Amines
Wurz, Ryan P.,Charette, Andre B.
, p. 1262 - 1269 (2007/10/03)
A practical synthesis for the preparation of a diverse series of cyclopropane α-amino acids is described. Nitrocyclopropane carboxylates can be readily prepared through treatment of α-nitroesters and iodobenzene diacetate or α-nitro-α-diazoesters with a R