292822-52-7Relevant articles and documents
2′-substituted analogs of cocaine: Synthesis and dopamine transporter binding potencies
El-Moselhy, Tarek F.,Avor, Kwasi S.,Basmadjian, Garo P.
, p. 275 - 278 (2001)
A series of 2′-substituted cocaine analogs (4-8) was prepared and evaluated in an in vitro dopamine transporter (DAT) binding assay. Compounds 4-7 were prepared by esterifying the 3β-hydroxyl group of ecgonine methyl ester (3) using the appropriate acid c