349639-42-5Relevant articles and documents
Synthesis of 3-amino-substituted N-alkylindazoles via palladium(II)- catalyzed intramolecular N-arylation of tosylhydrazines
Suryakiran,Prabhakar,Venkateswarlu
, p. 1370 - 1371 (2007)
An efficient synthesis of 3-amino-substituted N-alkyl indazoles is described. Reaction of readily available o-halo aryl hydrazines with palladium(II) acetate and cupper(I) iodide in the presence of a base afforded the corresponding 3-substituted N-tosylin
COMPOUNDS HAVING 5-HT6 RECEPTOR AFFINITY
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Page/Page column 114, (2010/11/28)
The present disclosure provides compounds having affinity for the 5HT6 receptor which are of the formula (I), wherein R1-R3 A, B, D, E, G, Q, and x are as defined herein. The disclosure also relates to methods of preparing such compounds, compositions containing such compounds, and methods of use thereof.