473918-47-7Relevant articles and documents
The copper-catalyzed N-arylation of indoles
Antilla, Jon C.,Klapars, Artis,Buchwald, Stephen L.
, p. 11684 - 11688 (2002)
A general method for the N-arylation of indoles using catalysts derived from Cul and trans-1,2-cyclohexanediamine (1a), trans-N,N′-dimethyl-1,2-cyclohexanediamine (2a), or N,N′-dimethyl-ethylenediamine (3) is reported. N-Arylindoles can be produced in high yield from the coupling of an aryl iodide or aryl bromide with a variety of indoles.