5180-75-6Relevant articles and documents
Design and development of novel p-aminobenzoic acid derivatives as potential cholinesterase inhibitors for the treatment of Alzheimer's disease
Shrivastava, Sushant K.,Sinha, Saurabh K.,Srivastava, Pavan,Tripathi, Prabhash N.,Sharma, Piyoosh,Tripathi, Manish K.,Tripathi, Avanish,Choubey, Priyanka K.,Waiker, Digambar K.,Aggarwal, Lalit M.,Dixit, Manish,Kheruka, Subhash C.,Gambhir, Sanjay,Shankar, Sharmila,Srivastava, Rakesh K.
, p. 211 - 223 (2019)
Based on the quantitative structure-activity relationship (QSAR), some novel p-aminobenzoic acid derivatives as promising cholinesterase enzyme inhibitors were designed, synthesized, characterized and evaluated to enhance learning and memory. The in vitro
Synthesis, analysis, cholinesterase-inhibiting activity and molecular modelling studies of 3-(dialkylamino)-2-hydroxypropyl 4-[(alkoxy-carbonyl)amino]benzoates and their quaternary ammonium salts
Padrtova, Tereza,Marvanova, Pavlina,Odehnalova, Klara,Kubinova, Renata,Parravicini, Oscar,Garro, Adriana,Enriz, Ricardo D.,Humpa, Otakar,Oravec, Michal,Mokry, Petr
, (2017/12/05)
Tertiary amines 3-(dialkylamino)-2-hydroxypropyl 4-[(alkoxycarbonyl)amino]benzoates and their quaternary ammonium salts were synthesized. The final step of synthesis of quaternary ammonium salts was carried out by microwave-assisted synthesis. Software-ca
Oxime-Based carbonates as useful reagents for both n-protection and peptide coupling
Jad, Yahya El-Sayed,Khattab, Sherine N.,El-Faham, Ayman,Albericio, Fernando
, p. 14361 - 14376 (2013/03/13)
We have demonstrated that oxime-based mixed carbonates are very effective reagents for both N-protection and peptide coupling.