54042-83-0Relevant articles and documents
Pharmaceutical compositions containing a 3-(amino-methylene)-5-phenyl-1,4-benzodiazepin-2-one and method of use
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, (2008/06/13)
Pharmaceutical dosage unit compositions containing as an active ingredient a compound of the formula SPC1 Wherein R1 and R2, which may be identical to or different from each other, are each hydrogen, cycloalkyl, phenyl, --A--Y wherein A is alkyl of 1 to 5 carbon atoms or alkenyl of 1 to 5 carbon atoms, and Y is furyl, dialkylamino, hydroxyl, carbalkoxy or carbamido, Or, together with each other and the nitrogen atom to which they are attached, pyrrolidino, piperidino, hexamethyleneimino, morpholino, thiomorpholino, thiomorpholino-S-oxide or N'-alkylpiperazino, R3 is halogen, nitro or trifluoromethyl, R4 is hydrogen, halogen or trifluoromethyl, and R5 is hydrogen, alkyl, cycloalkyl-methyl, alkylamino-alkyl, dialkylamino-alkyl or trifluoromethyl-alkyl; And a method of using the same as sedatives, tranquilizers, muscle-relaxants and anticonvulsives.