66636-17-7Relevant articles and documents
Evaluation of new benzimidazole derivatives as cysticidal agents: In vitro, in vivo and docking studies
González-Hernández, Iliana,Palomares-Alonso, Francisca,Becerril-Vega, José,De La Torre, Silvia Melchor-Doncel,Hernández-Luis, Francisco,Rodriguez-Morales, Sergio,Aguayo-Ortiz, Rodrigo,Dominguez, Laura,Rodríguez-Balderas, César A.,González-Maciel, Angélica,Rojas-Tomé, Irma Susana,Castro, Nelly,Jung-Cook, Helgi
, p. 1293 - 1300 (2019)
Based on our previous research on cysticidal drugs, we report the synthesis and evaluation of three new benzimidazole derivatives. In these compounds, the amido group was used as a bioisosteric replacement of the ester group. The molecular docking on β-tu
Removable saccharide-benzimidazole (BIM) tags and conjugates thereof via 1H-position of the benzimidazoles
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Page/Page column 17, (2015/07/27)
Novel method and reagents for generating reversibly tagged saccharides, aldehydes, carboxyl acids, or orthoacetates useful in analytical and diagnostic applications are disclosed. Saccharides are coupled at the reducing end to tagging moieties comprising
An efficient and highly chemoselective N-Boc protection of amines, amino acids, and peptides under heterogeneous conditions
Jahani, Fatemeh,Tajbakhsh, Mahmood,Khaksar, Samad,Azizi, Mohamad Reza
experimental part, p. 1035 - 1043 (2012/07/27)
A simple and efficient procedure for chemoselective mono-N-Boc protection of various structurally diverse amines, amino acids, and peptides with di-tert-butyl dicarbonate using Amberlyst-15 as catalyst in ethanol is described. The catalyst can be readily separated from the reaction products with simple filtration and recovered for direct reuse. No competitive side-reactions such as formation of isocyanate, urea, oxazolidinone, and N,N-di-Boc derivatives were observed.
