73841-41-5Relevant articles and documents
An intra/intermolecular suzuki sequence to benzopyridyloxepines containing geometrically pure exocyclic tetrasubstituted alkenes
Carson, Matthew W.,Giese, Matthew W.,Coghlan, Michael J.
supporting information; experimental part, p. 2701 - 2704 (2009/05/26)
(Chemical Equation Presented) A route to enable the preparation of 5-benzylidenyl-benzopyridyloxepine analogues was developed to continue our research in the field of nuclear hormone receptor modulators. The key steps are1) a syn-stereoselective diboratio
PIPERAZINE HETEROARYL DERIVATES AS GPR38 AGONISTS
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Page/Page column 39, (2010/11/25)
The invention provides compounds of formula (I) or pharmaceutically acceptable salts thereof, (I) wherein R1, R2, R3, R4, R5, R6, Z, X and B are as defined in the specification. The compounds are partial or full agonists at the GPR38 receptor. Pharmaceutical compositions comprising the compounds, methods of preparing the compounds, uses of the compounds and methods involving the compounds are also provided.
ADAMANTYL DERIVATES AS P2X7 RECEPTOR ANTAGONISTS
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Page/Page column 120-121, (2010/10/20)
The invention provides compounds of formula (I) pharmaceutically acceptable salt or solvate thereof, in which R1, A1, m and A are as defined in the specification; a process for their preparation; pharmaceutical compositions containin