79146-99-9Relevant articles and documents
Aminothiazoles and aminothiadiazoles as nucleophiles in aminocarbonylation of iodobenzene derivatives
Gergely, Máté,Kollár, László
, p. 2030 - 2040 (2018/03/21)
Various 2-, 3- and 4-substituted iodobenzenes were aminocarbonylated using aminothiazole and aminothiadiazole derivatives in palladium-catalysed reaction. The reaction is chemospecific toward the corresponding carboxamides. Consequently, the application o
Facile synthesis of N-acyl 2-aminobenzothiazoles by NHC-catalyzed direct oxidative amidation of aldehydes
Premaletha, Sethulekshmy,Ghosh, Arghya,Joseph, Sumi,Yetra, Santhivardhana Reddy,Biju, Akkattu T.
supporting information, p. 1478 - 1481 (2017/02/05)
A mild, general, and high yielding synthesis of N-acyl 2-aminobenzothiazoles has been demonstrated by N-heterocyclic carbene (NHC)-organocatalyzed direct amidation of aldehydes with 2-aminobenzothiazoles proceeding via acyl azolium intermediates. The carbene generated from the triazolium salt under oxidative conditions was the key for the success of this reaction. The method was subsequently applied to the synthesis of various biologically important N-acyl 2-aminobenzothiazoles.
Mesoionic purinone analogues as inhibitors of cyclic-AMP phosphodiesterase: A comparison of several ring systems
Rogers,Glennon,Smith,Boots,Nanavati,Maconaughey,Aub,Thomas,Bass,Mbagwu
, p. 1284 - 1287 (2007/10/02)
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