81336-57-4Relevant articles and documents
NOVEL PREPARATION METHOD OF QUINOLINE N-OXIDE DERIVATIVE WITH AMIDE GROUP
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Paragraph 138; 139, (2015/11/09)
Provided are a preparation method of a quinoline N-oxide derivative with an amide group capable of easily introducing the amide group into the quinoline N-oxide derivative by simplified processes and mild reaction conditions, and a quinoline N-oxide derivative with an amide group prepared by using the same.
A mild palladium-catalyzed Suzuki coupling reaction of quinoline carboxylates with boronic acids
Li, Wenjie,Gao, Joe J.,Zhang, Yongda,Tang, Wenjun,Lee, Heewon,Fandrick, Keith R.,Lu, Bruce,Senanayake, Chris H.
supporting information; experimental part, p. 1671 - 1675 (2011/09/20)
A palladium-catalyzed cross-coupling between aryl carboxylates and boronic acids has been achieved for the first time by taking advantage of the enhanced reactivity of quinoline 4-carboxylates. Also for the first time a Suzuki coupling reaction via a self-activation of boronic acids without addition of base is described. The reactions proceed under mild conditions (25-65°C) to give excellent yields, and a wide range of functionalities is tolerated. Copyright