917080-08-1Relevant articles and documents
TRICYCLIC COMPOUNDS AS HISTONE METHYL-TRANSFERASE INHIBITORS
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Page/Page column 162; 163, (2019/03/05)
The present disclosure provides certain tricyclic compounds that are histone methyltransferases G9a and/or GLP inhibitors and are therefore useful for the treatment of diseases treatable by inhibition of G9a and/or GLP such as cancers and hemoglobinopathi
Synthesis of 1-aryl-1H-indole derivatives by iodine-mediated cyclization of 2-(arylamino)styrene derivatives
Kobayashi, Kazuhiro,Miyamoto, Kazuna,Yamase, Tohru,Nakamura, Daizo,Morikawa, Osamu,Konishi, Hisatoshi
, p. 1580 - 1584 (2007/10/03)
A convenient synthetic method for 1-aryl-1H-indole derivatives has been developed. 2-(Arylamino)-α-methylstyrene derivatives were treated with iodine in the presence of sodium hydrogencarbonate to give 1-aryl-3-methyl-1H- indole derivatives in fair to goo