946488-41-1Relevant articles and documents
Exploration of a new series of CCR5 antagonists: Multi-dimensional optimization of a sub-series containing N-substituted pyrazoles
Lemoine, Remy C.,Petersen, Ann C.,Setti, Lina,Jekle, Andreas,Heilek, Gabrielle,Derosier, Andre,Ji, Changhua,Berry, Pamela,Rotstein, David M.
scheme or table, p. 4753 - 4756 (2010/10/02)
The introduction of N-substituted pyrazoles in a new series of CCR5 antagonists was shown to substantially increase antiviral activity.