95898-97-8Relevant articles and documents
FUSED [1,2,4]THIADIAZINE DERIVATIVES WHICH ACT AS KAT INHIBITORS OF THE MYST FAMILY
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Page/Page column 90, (2019/03/17)
A compound of formula (I): which inhibits the activity of one or more KATs of the MYST family, i.e., TIP60, KAT6B, MOZ, HBO1 and MOF.
THIAZOLYL COMPOUNDS USEFUL AS KINASE INHIBITORS
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Page/Page column 33, (2010/03/31)
The invention provides compounds of formula I [INSERT CHEMICAL STRUCTURE HERE] (I) and pharmaceutically acceptable salts thereof. The formula I thiazolyl compounds inhibit tyrosine kinase activity thereby making them useful as anticancer agents and for the treatment of Alzheimer's Disease.
Synthesis of N-methyl-4-pyridyl-1,2,3,4-tetrahydroisoquinolines via a Pictet-Spengler cyclisation
Prat,Bureau,Daveu,Levacher,Dupas,Queguiner,Bourguignon
, p. 767 - 771 (2007/10/03)
The synthesis of N-methyl-4-pyridyl-1,2,3,4-tetrahydroisoquinolines (6a,b,c) was achieved via a Pictet-Spengler cyclization of an activated amino group derivatized in a carbamate form. The obtained compounds have been designed as potential serotonin analo