HIGHLY FUNCTIONALIZED AZIRIDINES II: A FACILE SYNTHESIS OF DIETHYL AZIRIDINYLPHOSPHONATES AND 2-CHLOROAZIRIDINYLPHOSPHONATES
The reaction of diethyl 1-lithio-1-chloromethylphosphonate with aromatic imines gave aziridinylphosphonates in good yields and with an high stereoselectivity.The resulting aziridines reacted with n-BuLi and led to the 2-lithiated anions which were trapped with carbon tetrachloride to give 2-chloroaziridinylphosphonates in excellent yields.
Coutrot, Philippe,Elgadi, Abdelaziz,Grison, Claude
p. 1179 - 1192
(2007/10/02)
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