- DECONSTRUCTIVE FUNCTIONALIZATION METHODS AND COMPOUNDS
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Disclosed herein, inter alia, are deconstructive functionalization methods and compounds made using the same.
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Paragraph 0464-0467
(2020/01/31)
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- Rapid Assembly of Saturated Nitrogen Heterocycles in One-Pot: Diazo-Heterocycle “Stitching” by N–H Insertion and Cyclization
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Methods that provide rapid access to new heterocyclic structures in biologically relevant chemical space provide important opportunities in drug discovery. Here, a strategy is described for the preparation of 2,2-disubstituted azetidines, pyrrolidines, pi
- Boddy, Alexander J.,Affron, Dominic P.,Cordier, Christopher J.,Rivers, Emma L.,Spivey, Alan C.,Bull, James A.
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supporting information
p. 1458 - 1462
(2019/01/04)
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- ORGANIC COMPOUNDS
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A compound of formula (I) or tautomers, or stereoisomers, or solvates, or pharmaceutically acceptable salts thereof, wherein M1, M1, L1, L2, W1, W2, X1, X2, Y1, Y2, A, R5 and R5a are as defined herein for the for treatment of conditions mediated by the blockade of an epithelial sodium channel, particularly an inflammatory or allergic condition.
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Page/Page column 134
(2008/06/13)
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- CHEMICAL COMPOUNDS
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The present invention provides novel compounds that demonstrate protective effects on target cells from HIV infection in a manner as to bind specifically to the chemokine receptor, and which affect the binding of the natural ligand or chemokine to a receptor such as CXCR4 and/or CCR5 of a target cell.
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Page/Page column 78
(2010/10/20)
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- Malonic acid derivatives and methods for their synthesis
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The present invention refers to a new class of malonic acid derivatives of general formula I STR1 wherein R1 and R2, each independently, represent hydrogen or a carboxyl protecting group, and the residue R corresponds to the side-cha
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