European Journal of Medicinal Chemistry (2020)
Update date:2022-08-30
Topics:
Chen, Jianjun
Deng, Xin
Li, Gang
Li, Ling
Liu, Jin
Liu, Shuwen
Luo, Meihua
Ren, Yichang
Wang, Wei
Wang, Yuxi
A series of Pyrazolo[1,5-a]Pyrimidine analogs were designed and synthesized as novel tubulin inhibitors. Among them, compounds 1a and 1b showed the highest antiproliferative activity against a panel of cancer cell lines with average IC50 values
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