10.1002/anie.201704092
Angewandte Chemie International Edition
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[13] CCDC-1544647 (3be) contain the supplementary crystallographic data
for this paper. These data can be obtained free of charge from The
[6]
Cambridge
Crystallographic
Data
Centre
via
[14] The simple amine addition product underwent bromination with NBS to
give the expected product (shown for 3ae) in 40% isolated yield which
indicates that the suggested enolate does not necessarily has to be
generated during ring-opening (direct intramolecular proton-transfer).
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