107572-53-2Relevant articles and documents
An efficient 3-acylquinoline synthesis from acetophenones and anthranil: Via C(sp3)-H bond activation mediated by Selectfluor
Gao, Yejun,Hider, Robert C.,Ma, Yongmin
, p. 10340 - 10344 (2019/04/10)
An efficient method for the synthesis of 3-functionalized quinolines from commercially available acetophenones and anthranil has been described. Selectfluor propels the C(sp3)-H bond activation of the acetophenones and aza-Michael addition of anthranil resulting in annulated 3-acylquinolines in moderate to high yields. DMSO acts not only as a solvent but also as a one carbon donor in the reaction.
Synthesizing method of aromatic pyridinopyridine compound
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Paragraph 0084; 0085; 0086, (2017/07/20)
The invention discloses a synthesizing method of an aromatic pyridinopyridine compound, and belongs to the technical field of organic synthesizing. According to the technical scheme, the characteristics of the synthesizing method refers to the description. The method is simple, efficient, convenient to operate, mild in conditions, and wide in substrate applying scope.
Reaction of α-oxoketene-N,S-arylaminoacetals with Vilsmeier reagents: An efficient route to highly functionalized quinolines and their benzo/hetero-fused analogues
Mahata,Venkatesh,Syam Kumar,Ila,Junjappa
, p. 3966 - 3975 (2007/10/03)
A simple, highly efficient, and regioselective synthesis of functionalized quinolines through Vilsmeier cyclization of a variety of α-oxoketene-N,S-anilinoacetals has been reported. The cyclization is found to be facile with N,S-acetals bearing strongly a
