147688-34-4Relevant articles and documents
Orthogonal regioselective synthesis of N-alkyl-3-substituted tetrahydroindazolones
Kim, Jonghoon,Song, Heebum,Park, Seung Bum
supporting information; experimental part, p. 3815 - 3822 (2010/09/10)
A divergent strategy for the regioselective and orthogonal synthesis of complementary regioisomers of N-alkyl-3-substituted-tetrahydroindazolones 3 and 4 was achieved from. Boc-protected alkylhydrazmes 1. The robustness and sub-strate generality of this method were validated by synthesizing 3 and. 4 through the intra- and intermolecular condensation of 1 with various 2-acylcyclohexane-l,3-diones 2 and aldehydes, respectively.
Pyrazolones as inhibitors of 11B-hydroxysteroid dehydrogenase
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Page/Page column 25, (2008/06/13)
Provided herein are compounds of the formula (I): as well as pharmaceutically acceptable salts thereof, wherein the substituents are as those disclosed in the specification. These compounds, and the pharmaceutical compositions containing them, are useful for the treatment of diseases such as, for example, type II diabetes mellitus and metabolic syndrome.
N-tert-butoxycarbonylaminophthalimide, a versatile reagent for the conversion of alcohols into alkylated tert-butylcarbazates or hydrazines via the Mitsunobu protocol
Brosse, Nicolas,Pinto, Maria-Fatima,Jamart-Grégoire, Brigitte
, p. 205 - 207 (2007/10/03)
An efficient two-step method has been developed for the conversion of alcohols to substituted hydrazines. The use of N-tert- butoxycarbonylaminophthalimide as an acid partner in Mitsunobu reactions with a variety of alcohols permits the synthesis of the corresponding monoalkylated tert-butylcarbazates and hydrazines.