1610362-87-2Relevant articles and documents
Fluorescence polarization for the evaluation of small-molecule inhibitors of PCAF BRD/Tat-AcK50 association
Hu, Ping,Wang, Xinghui,Zhang, Baiqun,Zhang, Shuai,Wang, Qiang,Wang, Zhiyong
supporting information, p. 928 - 931 (2014/05/20)
A fluorescence polarization competitive assay was developed to efficiently screen and evaluate inhibitors of PCAF bromodomain/Tat-AcK50 protein-peptide interaction. A series of pyridine 1-oxide derivatives were synthesized and evaluated. Some of the novel