256381-13-2Relevant articles and documents
NRF2 ACTIVATOR
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Page/Page column 113; 116, (2018/08/20)
Provided are tetrahydroisoquinoline derivatives as Nrf2 activators.
Synthesis, biological evaluation and molecular modelling of sulfonohydrazides as selective PI3K p110α inhibitors
Kendall, Jackie D.,Rewcastle, Gordon W.,Frederick, Raphael,Mawson, Claire,Denny, William A.,Marshall, Elaine S.,Baguley, Bruce C.,Chaussade, Claire,Jackson, Shaun P.,Shepherd, Peter R.
, p. 7677 - 7687 (2008/03/14)
A series of 2-methyl-5-nitrobenzenesulfonohydrazides were prepared and evaluated as inhibitors of PI3K. An isoquinoline derivative shows good selectivity for the p110α isoform over p110β and p110δ, and also demonstrates good in vitro activity in a cell pr
Biarylpropylsulfonamides as novel, potent potentiators of 2-amino-3-(5-methyl-3-hydroxyisoxazol-4-yl)-propanoic acid (AMPA) receptors [1]
Ornstein,Zimmerman,Arnold,Bleisch,Cantrell,Simon,Zarrinmayeh,Baker,Gates,Tizzano,Bleakman,Mandelzys,Jarvie,Ho,Deverill,Kamboj
, p. 4354 - 4358 (2007/10/03)
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