56347-09-2Relevant articles and documents
Pd-catalyzed Suzuki/Sonogashira cross-coupling reaction and the direct sp3 arylation of 7-chloro-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidine
Loubidi, Mohammed,Moutardier, Ana?s,Campos, Joana F.,Berteina-Raboin, Sabine
, p. 1050 - 1054 (2018)
A rapid and efficient method is reported for the synthesis of the [1,2,4]triazolo[1,5-a]pyrimidine motif. Palladium catalyzed Suzuki and Sonogashira cross coupling reactions on 7-chloro-5-methyl-[1,2,4]triazolo[1,5-a]pyrimidine were performed. The direct sp3 arylation of compounds resulting from the Suzuki reaction was then carried out.
CHEMICAL CONVERSIONS OF 5,7-DISUBSTITUTED DIHYDRO-1,2,4-TRIAZOLOPYRIMIDINES
Desenko, S. M.,Orlov, V. D.,Lipson, V. V.
, p. 1362 - 1366 (2007/10/02)
Hydrolysis, oxidation, reduction, alkylation, and nitrosation of aromatic-substituted dihydro-1,2,4-triazolopyrimidines have been studied.