60987-18-0Relevant articles and documents
Ligands for the common allosteric site of acetylcholine M2-receptors: Development and application
Holzgrabe,Bender,Botero Cid,Staudt,Pick,Pfletschinger,Balatkova,Traenkle,Mohr
, p. 149 - 155 (2000)
Ligands for the allosteric site of acetylcholine M2 receptors are able to retard the dissociation of simultaneously bound ligands for the orthosteric site. This effect promotes receptor occupation by the orthosteric ligand. The allosteric effec