76413-56-4Relevant articles and documents
Peptide-bond Formation, Chemoselective Acylation of Amino Acids, and Crosslinking Reaction between Amino Acids Utilizing a Functional Five-membered Heterocycle, 1,3-Thiazolidine-2-thione
Nagao, Yoshimitsu,Miyasaka, Tadayo,Seno, Kaoru,Fujita, Eiichi,Shibata, Daisuke,Doi, Etsushiro
, p. 2439 - 2446 (2007/10/02)
The monitored aminolysis of 3-acyl-1,3-thiazolidine-2-thiones has been extended to the peptide-bond formation, the chemoselective acylation of amino acids having multifunctional groups, and the crosslinking reaction between amino acids.
Studies on Peptides. XCIV. Thiazoline-2-thione as a Carboxyl-activating Reagent for Peptide Synthesis
Yajima, Haruaki,Akaji, Kenichi,Hirota, Yoriko,Fujii, Nobutaka
, p. 3140 - 3142 (2007/10/02)
3-Acyl derivatives obtained from the DCC condensation of Nα-protected amino acids and thiazoline-2-thione were found to be useful for peptide synthesis, in the same way as active esters.Keywords---3-acylthiazoline-2-thione derivatives of N