58202-26-9Relevant articles and documents
Design, synthesis and biological activities of dihydroaurones
VENKATESWARLU, SOMEPALLI,MURTY, GANDROTU NARASIMHA,SATYANARAYANA, MEKA,SIDDAIAH, VIDAVALUR
, p. 1396 - 1402 (2021/06/09)
To widen aurones applicability in achromatic food and cosmetic applications, a series of dihydroaurones were designed to mimic natural aurones as well as synthetic aurones. Dihydroaurones have been synthesized from the corresponding aurones by hydrogenation. These dihydroaurones and their corresponding aurones were screened for antioxidant, anti-inflammatory and tyrosinase enzyme inhibitory activity. Synthesized dihydroaurones (3b-f) displayed superior antioxidant activity in superoxide free radical scavenging assay than the standard gallic acid. Dihydroaurones (3b-f) also exhibited significant tyrosinase enzyme inhibitory activity and two dihydroaurones (3h, 3j) showed promising 5-lipoxygenase inhibitory activity.
Synthesis and structure-affinity-activity relationships of novel benzofuran derivatives as MT2 melatonin receptor selective ligands
Wallez, Valérie,Durieux-Poissonnier, Sophie,Chavatte, Philippe,Boutin, Jean A.,Audinot, Valérie,Nicolas, Jean-Paul,Bennejean, Caroline,Delagrange, Philippe,Renard, Pierre,Lesieur, Daniel
, p. 2788 - 2800 (2007/10/03)
A series of N-(2-phenylbenzofuran-3-yl) ethyl amide and N-(2-arylalkylbenzofuran-3-yl) ethyl amide derivatives were synthesized and evaluated as melatonin receptor ligands. The affinity of each compound for the two MT1 and MT2 melato
The Stevens -Shift of Oxonium Ylides: A Route to Substituted Tetrahydrofuranones
Eberlein, T. H.,West, F. G.,Tester, R. W.
, p. 3479 - 3482 (2007/10/02)
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